| Saturday, September 19, 2009 | ||
| 08:00:00 | Introduction | |
| 08:05:00 | Nature Chemical Biology | |
| 08:10:00 | What does chemical biology have to offer and what does drug development need? | Paul Workman |
| 08:35:00 | Cell-based screening and target deconvolution | |
| 08:40:00 | Session chair: | Gerard Drewes |
| 08:50:00 | The gap between scientists' aspirations and society's expectations | Stuart Schreiber |
| 09:30:00 | A combined chemical genetic/RNAi approach: New tools to study cell division | Ulrike Eggert |
| 10:10:00 | Knowledge-based triaging of chemical biology screens | Jeremy Jenkins |
| 10:50:00 | Coffee Break | |
| 10:50:00 | Genomic information in drug discovery | Todd Golub |
| 11:10:00 | Chemical genomic tools to understand drug action and gene function | Guri Giaever |
| 12:00:00 | Systems biology from drug combinations | Joseph Lehar |
| 12:30:00 | Lunch | |
| 12:35:00 | Targeting pathways and systems | |
| 13:30:00 | Session chair: | Carolyn Cho |
| 13:40:00 | Chemical proteomics and the mechanism of action of kinase inhibitors | Giulio Superti-Furga |
| 15:00:00 | The chemical biology of behavior and psychiatric disease | Randall Peterson |
| 15:40:00 | Coffee Break | |
| 16:10:00 | A systems biology approach to the discovery of novel pathways | Cristiano Migliorini |
| 16:50:00 | Do system biologists need robot chemists? | Andrew Hopkins |
| 17:30:00 | Reception and Poster Session | |
| 17:35:00 | Announcements | |
| Sunday, September 20, 2009 | ||
| 08:25:00 | Expanding druggable chemical space | |
| 08:30:00 | Session chair: | Michael Hannus |
| 08:40:00 | Exploration of chemical space for drug discovery by database generation | Jean-Louis Reymond |
| 09:20:00 | Thinking the undruggable: Peptides, peptidomimetics, and natural products | Peter Wipf |
| 10:00:00 | Alkaloid biosynthesis in periwinkle | Sarah O'Connor |
| 10:40:00 | Coffee Break | |
| 11:10:00 | Natural product-based libraries for chemical biology and drug discovery | Derek Tan |
| 11:50:00 | Figments, fragments, and the gobsmacking emptiness of chemical space | Brian K Shoichet |
| 12:30:00 | Lunch | |
| 12:35:00 | Expanding druggable targets | |
| 13:30:00 | Session chair: | Stephen Fesik |
| 13:40:00 | Chemical genetic dissection of protein and lipid kinase regulatory networks | Kevan M Shokat |
| 14:40:00 | Oxygenase mediated epigenetic modifications - emerging targets for drug discovery | Christopher Schofield |
| 15:00:00 | Targeting cancer pathways with small molecule kinase inhibitors | Nathanael Gray |
| 15:40:00 | Coffee Break | |
| 16:10:00 | Drug discovery harnessing RNA interference | |
| 16:50:00 | Drugging the "undruggable" | Gregory Verdine |