3D Tissue Models
Inaugural Fragment-Based Techniques
1775 East Mission Bay Drive
San Diego, CA 92109
Inaugural  Fragment-Based Techniques
Cambridge Healthtech Institute

Schedule of Presentations:

Tuesday, April 7, 2009
12:30:00 Registration
13:30:00 Chairperson’s Opening Remarks Yoshitomo Hamuro
13:40:00 Fragment- Based Drug Design by Amide Hydrogen/Deuterium Exchange Mass Spectrometry Yoshitomo Hamuro
14:10:00 Native Mass Spectrometry: An ESI Tool for Fragment Library Screening Denis Zeyer
14:40:00 Use of SPR for Fragment Screening, HTS Hit Validation, and SAR Support in Drug Discovery Tony M. Giannetti
15:10:00 Screening of a Metabolite-Based Fragment Library Using X-ray Crystallography and SPR Alex Burgin
15:25:00 Networking Refreshment Break in the Exhibit Hall
16:05:00 Experimental Design in SPR Biosensor-based Fragment Screening Peer Källblad
16:35:00 Use of SPR for Protein-Nucleic Acid Interactions Farid Ahmed
17:05:00 Breakout Discussions with the Experts
17:10:00 Topic 1: SPR – what we need to know Peer Källblad
17:15:00 Topic 3: How to choose the right fragments to move forward Tony M. Giannetti
17:15:00 Topic 2: Selecting the right tools – what works? Denis Zeyer
18:15:00 End of Day
Wednesday, April 8, 2009
07:45:00 Morning Coffee
08:15:00 Chairperson’s Remarks Marcel Verdonk
08:20:00 Perspectives on NMR in Drug Discovery: a Technique Comes of Age KEYNOTE PRESENTATION Maurizio Pellecchia
09:00:00 Breakout Discussion Feedback by Moderators
09:30:00 Target Immobilization Provides New Opportunities in NMR-Based Fragment Discovery and Characterization Gregg Siegal
10:00:00 Networking Coffee Break in the Exhibit Hall
10:45:00 Docking and Scoring of Fragments Marcel Verdonk
11:15:00 Highly Efficient Screening Technology for the Selection of Fragments for X-Ray Crystallography Doris Hafenbradl
11:45:00 Target-Tailored Ligand Databases for Virtual Screening Bogdan Iorga
12:15:00 Walk and Talk Luncheon in the Exhibit Hall (Last Chance for Exhibit Viewing)
13:55:00 Chairperson’s Remarks Gregg Siegal
14:00:00 Chemotyping and Fragment Based Drug Design Hugo O. Villar
14:30:00 Enzymatic Assays for Fragment-Based Screening using Enthalpy Array Technology Michael I. Recht
15:00:00 Networking Refreshment Break
15:20:00 Fragment Library Screening: from Virtual Screening of Chemical Space to Rapid Candidate Nomination David Bailey
15:50:00 Unprecedented Natural Product Scaffolds as the Basis of a Fragment Based Screening Library Dmitry Genis
16:20:00 Panel Discussion: Fragment-based Drug Discovery – integrating library screening strategies to deliver novel candidates David Bailey
16:50:00 End of Conference
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